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Approved focused synthesisEvidence current through August 2026

MRI-Measured Liver Fat in the LY3437943 Phase 2 Substudy

September 01, 2026 · 4 minutes

Investigators reported striking liver-fat changes in a randomized LY3437943 substudy—one of the most closely watched findings outside the primary body-weight and glycemic endpoints. The study offers a strong signal for imaging-defined steatosis and a clear rationale for dedicated liver research.

Evidence boundary: Liver findings below come from a prespecified MRI substudy of Lilly’s investigated LY3437943. They are imaging results under that protocol, not claims about another material or a recommended use.

Investigators reported striking liver-fat changes in a randomized LY3437943 substudy—one of the most closely watched findings outside the primary body-weight and glycemic endpoints. The study offers a strong signal for imaging-defined steatosis and a clear rationale for dedicated liver research.

The MRI-PDFF substudy

A prespecified substudy enrolled 98 participants from the Phase 2 obesity trial who had sufficient liver fat at baseline. At week 24, relative liver-fat changes were approximately:

Group Relative liver-fat change
Lower dose −42.9%
Intermediate dose −57.0%
Higher dose −81.4%
Highest dose −82.4%
Placebo +0.3%

Imaging-defined liver-fat normalization below 5% occurred in 27%, 52%, 79%, and 86% of the retatrutide groups, compared with 0% for placebo.

These are large randomized imaging findings.

Why imaging is not the entire disease

MRI-PDFF quantifies hepatic fat. It does not directly show hepatocyte injury, inflammation, ballooning, fibrosis stage, cirrhosis progression, decompensation, transplantation, or mortality.

The substudy did not include liver biopsies. FIB-4 and enhanced liver fibrosis measures did not improve consistently, and the analyses were not multiplicity adjusted. Therefore, the evidence did not establish histologic steatohepatitis resolution or fibrosis regression.

What may explain the change?

Substantial weight loss commonly reduces liver fat. Retatrutide’s receptor profile could also contribute through metabolic mechanisms, but this substudy could not isolate a weight-independent effect or assign the result to the glucagon receptor.

Dedicated liver trials and biopsy or clinical-outcome evidence are needed to answer those questions.

Bottom line

The LY3437943 evidence includes strong preliminary MRI findings, with many participants reaching the study’s imaging-defined liver-fat threshold. This is a meaningful result within the substudy. Biopsy-based and longer-term research will determine whether the observed imaging changes extend to inflammation, fibrosis, and clinical liver outcomes.

Study map

Study records discussed

Peer-reviewed human trials and related publicationsSee approved evidence mapCompleted

New England Journal of Medicine

RET-STUDY-P004

Jastreboff AM, et al. Triple-hormone-receptor agonist retatrutide for obesity. New England Journal of Medicine. 2023. DOI: 10.1056/NEJMoa2301972. PMID: 37366315. NCT04881760. https://doi.org/10.1056/NEJMoa2301972

View study
Peer-reviewed human trials and related publicationsSee approved evidence mapCompleted

Nature Medicine

RET-STUDY-P006

Sanyal AJ, et al. Retatrutide and liver fat in the Phase 2 obesity cohort. Nature Medicine. 2024. DOI: 10.1038/s41591-024-03018-2. PMID: 38858523. PMCID: PMC11271400. https://pmc.ncbi.nlm.nih.gov/articles/PMC11271400/

View study

Permanent sources

Reference ledger

  1. P004Peer-reviewed human trials and related publications

    New England Journal of Medicine

    Jastreboff AM, et al. Triple-hormone-receptor agonist retatrutide for obesity. Jastreboff AM, et al. Triple-hormone-receptor agonist retatrutide for obesity. New England Journal of Medicine. 2023. DOI: 10.1056/NEJMoa2301972. PMID: 37366315. NCT04881760. https://doi.org/10.1056/NEJMoa2301972(2023). DOI: 10.1056/NEJMoa2301972

  2. P006Peer-reviewed human trials and related publications

    Nature Medicine

    Sanyal AJ, et al. Retatrutide and liver fat in the Phase 2 obesity cohort. Sanyal AJ, et al. Retatrutide and liver fat in the Phase 2 obesity cohort. Nature Medicine. 2024. DOI: 10.1038/s41591-024-03018-2. PMID: 38858523. PMCID: PMC11271400. https://pmc.ncbi.nlm.nih.gov/articles/PMC11271400/(2024). DOI: 10.1038/s41591-024-03018-2

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